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Chemical structure of Histamine H4 receptor antagonist-1

GC70909

Histamine H4 receptor antagonist-1

Also known as 7-[2-amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-yl]-N-[(2S)-1-(dimethylamino)-1-oxo-3-phenylpropan-2-yl]-3,4-dihydro-1H-isoquinoline-2-carboxamide

Histamine H4 receptor antagonist-1 is an antagonist of histamine H4 receptor extracted from patent WO2010108059A1 compound 60

ChemicalCAS1246207-84-0MW542.68FormulaC30H38N8O2
CAS number
1246207-84-0
Molecular weight
542.68
Formula
C30H38N8O2
Solubility
DMSO ： 100 mg/mL (184·27 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
InChIKey
AVTPLFSHOMCNRC-SANMLTNESA-N
Catalogue number
GC70909
Brand
GLPBIO
Computed properties PubChem CID 59496678 · XLogP 2.5 · TPSA 111 Ų · H-bond donors 2
XLogP
2.5
TPSA
111 Ų
H-bond donors
2
H-bond acceptors
7
Rotatable bonds
6
Heavy atoms
40

SMILES CN1CCN(CC1)C2=NC(=NC(=C2)C3=CC4=C(CCN(C4)C(=O)N[C@@H](CC5=CC=CC=C5)C(=O)N(C)C)C=C3)N

Computed descriptors from PubChem (CID 59496678), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

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Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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