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Chemical structure of ENMD-2076 Tartrate

GC69068

ENMD-2076 Tartrate

Also known as (2R,3R)-2,3-dihydroxybutanedioic acid;6-(4-methylpiperazin-1-yl)-N-(5-methyl-1H-pyrazol-3-yl)-2-[(E)-2-phenylethenyl]pyrimidin-4-amine

ENMD-2076 Tartrate is a multi-target kinase inhibitor that inhibits Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, FGFR2, Src and PDGFRα with IC50 values of 1·86, 14, 58·2, 15·9, 92·7, 70·8 ,20·2 and 56·4 nM respectively

ChemicalCAS1453868-32-0MW525.56FormulaC25H31N7O6
CAS number
1453868-32-0
Molecular weight
525.56
Formula
C25H31N7O6
Solubility
DMSO ： 25 mg/mL (47·57 mM; Need ultrasonic)
InChIKey
KGWWHPZQLVVAPT-STTJLUEPSA-N
Catalogue number
GC69068
Brand
GLPBIO
Computed properties PubChem CID 24776050 · TPSA 188 Ų · H-bond donors 6 · H-bond acceptors 12
TPSA
188 Ų
H-bond donors
6
H-bond acceptors
12
Rotatable bonds
8
Heavy atoms
38

SMILES CC1=CC(=NN1)NC2=CC(=NC(=N2)/C=C/C3=CC=CC=C3)N4CCN(CC4)C.[C@@H]([C@H](C(=O)O)O)(C(=O)O)O

Computed descriptors from PubChem (CID 24776050), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.