GC65906
RXFP3/4 agonist 2
Also known as methyl 4-[2-[[amino-[(2E)-2-[(5-cyano-7-methyl-1H-indol-3-yl)methylidene]hydrazinyl]methylidene]amino]ethyl]benzoate
RXFP3/4 agonist 2 is a potent, nonpeptide dual RXFP3/4 agonist (EC50=3·1 and 2·7 nM)· RXFP3/4 agonist 2 also potently promotes interactions between RXFP3 and β-arrestin-2 with EC50 values in the range of 10-22 nM
ChemicalCAS2752378-78-0MW402.45FormulaC22H22N6O2
- CAS number
- 2752378-78-0
- Molecular weight
- 402.45
- Formula
- C22H22N6O2
- Solubility
- DMSO ： 100 mg/mL (248·48 mM; Need ultrasonic)
- InChIKey
- XIVYUSRYHWXGLX-UVHMKAGCSA-N
- Catalogue number
- GC65906
- Brand
- GLPBIO
Computed properties PubChem CID 162679305 · XLogP 2.7 · TPSA 129 Ų · H-bond donors 3
- XLogP
- 2.7
- TPSA
- 129 Ų
- H-bond donors
- 3
- H-bond acceptors
- 5
- Rotatable bonds
- 8
- Heavy atoms
- 30
SMILES CC1=CC(=CC2=C1NC=C2/C=N/NC(=NCCC3=CC=C(C=C3)C(=O)OC)N)C#N
Computed descriptors from PubChem (CID 162679305), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
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