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Chemical structure of GB-88

GC65439

GB-88

Also known as N-[(2S)-3-cyclohexyl-1-[[(2S,3S)-3-methyl-1-oxo-1-spiro[indene-1,4'-piperidine]-1'-ylpentan-2-yl]amino]-1-oxopropan-2-yl]-1,2-oxazole-5-carboxamide

GB-88 is an oral, selective non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 ?M

ChemicalCAS1416435-96-5MW546.7FormulaC32H42N4O4
CAS number
1416435-96-5
Molecular weight
546.7
Formula
C32H42N4O4
Solubility
DMSO ： 31·25 mg/mL (57·16 mM; Need ultrasonic)
InChIKey
DCUDDCGUKZLQLN-MCOVPRHSSA-N
Catalogue number
GC65439
Brand
GLPBIO
Computed properties PubChem CID 57330164 · XLogP 6.5 · TPSA 105 Ų · H-bond donors 2
XLogP
6.5
TPSA
105 Ų
H-bond donors
2
H-bond acceptors
5
Rotatable bonds
9
Heavy atoms
40

SMILES CC[C@H](C)[C@@H](C(=O)N1CCC2(CC1)C=CC3=CC=CC=C23)NC(=O)[C@H](CC4CCCCC4)NC(=O)C5=CC=NO5

Computed descriptors from PubChem (CID 57330164), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.