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Chemical structure of DRAK2-IN-1

GC65140

DRAK2-IN-1

Also known as N-[2-hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]pentanamide

DRAK2-IN-1, compound 16, is a potent, selective and ATP-competitive DRAK2 inhibitor with IC50and Kivalues of 3 nM and 0·26 nM, respectively

ChemicalCAS871837-60-4MW376.41FormulaC21H20N4O3
CAS number
871837-60-4
Molecular weight
376.41
Formula
C21H20N4O3
Solubility
DMSO ： 125 mg/mL (332·08 mM; Need ultrasonic)
InChIKey
ZFZLSKZDOULLMO-UHFFFAOYSA-N
Catalogue number
GC65140
Brand
GLPBIO
Computed properties PubChem CID 136175114 · XLogP 3.7 · TPSA 110 Ų · H-bond donors 4
XLogP
3.7
TPSA
110 Ų
H-bond donors
4
H-bond acceptors
4
Rotatable bonds
5
Heavy atoms
28

SMILES CCCCC(=O)NC1=CC2=C(C=C1)NC(=C2C3=C(C4=CC=CC=C4N3)N=O)O

Computed descriptors from PubChem (CID 136175114), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.