Loading...
Chemical structure of Bomedemstat

GC64865

Bomedemstat

Also known as N-[(2S)-5-[[(1R,2S)-2-(4-fluorophenyl)cyclopropyl]amino]-1-(4-methylpiperazin-1-yl)-1-oxopentan-2-yl]-4-(triazol-1-yl)benzamide

Bomedemstat (IMG-7289) is an orally active and irreversible lysine-specific demethylase 1 (LSD1) inhibitor· Bomedemstat can increase H3K4 and H3K9 methylation, and then alter gene expression· Bomedemstat shows anti-cancer activities, inhibits cancer cell proliferation and induces apoptosis

ChemicalCAS1990504-34-1MW519.61FormulaC28H34FN7O2
CAS number
1990504-34-1
Molecular weight
519.61
Formula
C28H34FN7O2
Solubility
DMSO ： 100 mg/mL (192·45 mM; Need ultrasonic)
InChIKey
KQKBMHGOHXOHTD-KKUQBAQOSA-N
Catalogue number
GC64865
Brand
GLPBIO
Computed properties PubChem CID 122460381 · XLogP 2.3 · TPSA 95.4 Ų · H-bond donors 2
XLogP
2.3
TPSA
95.4 Ų
H-bond donors
2
H-bond acceptors
7
Rotatable bonds
10
Heavy atoms
38

SMILES CN1CCN(CC1)C(=O)[C@H](CCCN[C@@H]2C[C@H]2C3=CC=C(C=C3)F)NC(=O)C4=CC=C(C=C4)N5C=CN=N5

Computed descriptors from PubChem (CID 122460381), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.