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Chemical structure of Bezuclastinib

GC64810

Bezuclastinib

Also known as 4,5-dimethyl-N-(2-phenyl-1H-pyrrolo[2,3-b]pyridin-5-yl)-1H-pyrazole-3-carboxamide

Bezuclastinib (CGT9486; PLX 9486) is a potent inhibitor of c-kit and c-kit D816V (0·0001＜IC50＜1 μM; extracted from patent WO2014100620 A2, compound P-2007)

ChemicalCAS1616385-51-3MW331.37FormulaC19H17N5O
CAS number
1616385-51-3
Molecular weight
331.37
Formula
C19H17N5O
InChIKey
NVSHVYGIYPBTEZ-UHFFFAOYSA-N
Catalogue number
GC64810
Brand
GLPBIO
Computed properties PubChem CID 75593308 · XLogP 3.2 · TPSA 86.5 Ų · H-bond donors 3
XLogP
3.2
TPSA
86.5 Ų
H-bond donors
3
H-bond acceptors
3
Rotatable bonds
3
Heavy atoms
25

SMILES CC1=C(NN=C1C(=O)NC2=CN=C3C(=C2)C=C(N3)C4=CC=CC=C4)C

Computed descriptors from PubChem (CID 75593308), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

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