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Chemical structure of Opiranserin hydrochloride

GC64690

Opiranserin hydrochloride

Also known as 4-butoxy-N-[[4-(dimethylamino)oxan-4-yl]methyl]-3,5-dimethoxybenzamide;hydrochloride

Opiranserin (VVZ-149) hydrochloride, a non-opioid and non-NSAID analgesic candidate, is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0·86 and 1·3 μM, respectively

ChemicalCAS1440796-75-7MW430.97FormulaC21H35ClN2O5
CAS number
1440796-75-7
Molecular weight
430.97
Formula
C21H35ClN2O5
Solubility
DMSO ： 50 mg/mL (116·02 mM; Need ultrasonic)
InChIKey
GSCGQHXDHYVKOL-UHFFFAOYSA-N
Catalogue number
GC64690
Brand
GLPBIO
Computed properties PubChem CID 71566777 · TPSA 69.3 Ų · H-bond donors 2 · H-bond acceptors 6
TPSA
69.3 Ų
H-bond donors
2
H-bond acceptors
6
Rotatable bonds
10
Heavy atoms
29

SMILES CCCCOC1=C(C=C(C=C1OC)C(=O)NCC2(CCOCC2)N(C)C)OC.Cl

Computed descriptors from PubChem (CID 71566777), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

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