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Chemical structure of Eliapixant

GC62950

Eliapixant

Also known as 3-(5-methyl-1,3-thiazol-2-yl)-5-[(3R)-oxolan-3-yl]oxy-N-[(1R)-1-[2-(trifluoromethyl)pyrimidin-5-yl]ethyl]benzamide

Eliapixant (BAY 1817080) is a potent and selective antagonist of P2X3 receptor, with an IC50 of 8 nM

ChemicalCAS1948229-21-7MW478.49FormulaC22H21F3N4O3S
CAS number
1948229-21-7
Molecular weight
478.49
Formula
C22H21F3N4O3S
Solubility
DMSO ： 33·33 mg/mL (69·66 mM; ultrasonic and warming and heat to 60°C)
InChIKey
GTQPEQGDLVSFJO-CXAGYDPISA-N
Catalogue number
GC62950
Brand
GLPBIO
Computed properties PubChem CID 121397587 · XLogP 3.4 · TPSA 114 Ų · H-bond donors 1
XLogP
3.4
TPSA
114 Ų
H-bond donors
1
H-bond acceptors
10
Rotatable bonds
6
Heavy atoms
33

SMILES CC1=CN=C(S1)C2=CC(=CC(=C2)O[C@@H]3CCOC3)C(=O)N[C@H](C)C4=CN=C(N=C4)C(F)(F)F

Computed descriptors from PubChem (CID 121397587), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.