GC62891
CCG258208 hydrochloride
CCG258208 (GRK2-IN-1) hydrochloride is a potent and selective GRK2 (G protein-coupled receptor kinase 2) inhibitor (IC50=30 nM) while maintaining 230-fold selectivity over GRK5 (IC50=7·09 μM) and more than 2500-fold selectivity over GRK1 (IC50=87·3 μM), PKA, and ROCK1
ChemicalMW488.94FormulaC24H26ClFN4O4
- CAS number
- —
- Molecular weight
- 488.94
- Formula
- C24H26ClFN4O4
- Solubility
- DMSO ： 250 mg/mL (511·31 mM; Need ultrasonic)|Water ： 50 mg/mL (102·26 mM; Need ultrasonic)
- Catalogue number
- GC62891
- Brand
- GLPBIO
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il