
GC62849
AS-99 TFA
AS-99 TFA is a first-in-class, potent and selective ASH1L histone methyltransferase inhibitor (IC50=?0·79??M, Kd=?0·89??M) with anti-leukemic activity· AS-99 TFA blocks cell proliferation, induces apoptosis and differentiation, downregulates MLL fusion target genes, and reduces the leukemia burden in vivo
ChemicalMW707.71FormulaC29H31F6N5O5S2
- CAS number
- —
- Molecular weight
- 707.71
- Formula
- C29H31F6N5O5S2
- Solubility
- DMSO : 250 mg/mL (353·25 mM; Need ultrasonic)
- Catalogue number
- GC62849
- Brand
- GLPBIO
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il