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Chemical structure of Ralaniten

GC62683

Ralaniten

Also known as (2R)-3-[4-[2-[4-[(2S)-3-chloro-2-hydroxypropoxy]phenyl]propan-2-yl]phenoxy]propane-1,2-diol

Ralaniten (EPI-002) is a potent and orally active antagonist of the androgen receptor-N-terminal domain (AR-NTD)· Ralaniten inhibits AR transcriptional activity, with IC50 of 7·4 μM· Ralaniten can be used for the research of castration-resistant prostate cancer (CRPC)

ChemicalCAS1203490-23-6MW394.89FormulaC21H27ClO5
CAS number
1203490-23-6
Molecular weight
394.89
Formula
C21H27ClO5
Solubility
DMSO ： 100 mg/mL (253·24 mM; Need ultrasonic)
InChIKey
HDTYUHNZRYZEEB-QZTJIDSGSA-N
Catalogue number
GC62683
Brand
GLPBIO
Computed properties PubChem CID 45107537 · XLogP 3.3 · TPSA 79.2 Ų · H-bond donors 3
XLogP
3.3
TPSA
79.2 Ų
H-bond donors
3
H-bond acceptors
5
Rotatable bonds
10
Heavy atoms
27

SMILES CC(C)(C1=CC=C(C=C1)OC[C@@H](CO)O)C2=CC=C(C=C2)OC[C@@H](CCl)O

Computed descriptors from PubChem (CID 45107537), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.