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Chemical structure of CPI-1612

GC62669

CPI-1612

Also known as (2R)-2-[[(2S)-2-(4-cyanophenyl)propyl]amino]-N-[5-(1-methylpyrazol-4-yl)-2-pyridinyl]-2-phenylacetamide

CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC50 of 8·1 nM for EP300 HAT· CPI-1612 has an anticancer activity

ChemicalCAS2374971-81-8MW450.53FormulaC27H26N6O
CAS number
2374971-81-8
Molecular weight
450.53
Formula
C27H26N6O
Solubility
DMSO ： 100 mg/mL (221·96 mM; Need ultrasonic)
InChIKey
SEDFZSHSBUXKAC-NIYFSFCBSA-N
Catalogue number
GC62669
Brand
GLPBIO
Computed properties PubChem CID 146014965 · XLogP 3.6 · TPSA 95.6 Ų · H-bond donors 2
XLogP
3.6
TPSA
95.6 Ų
H-bond donors
2
H-bond acceptors
5
Rotatable bonds
8
Heavy atoms
34

SMILES C[C@H](CN[C@H](C1=CC=CC=C1)C(=O)NC2=NC=C(C=C2)C3=CN(N=C3)C)C4=CC=C(C=C4)C#N

Computed descriptors from PubChem (CID 146014965), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
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Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.