GC61365
UPGL00004
Also known as 2-phenyl-N-[5-[[1-[5-[(2-phenylacetyl)amino]-1,3,4-thiadiazol-2-yl]piperidin-4-yl]amino]-1,3,4-thiadiazol-2-yl]acetamide
UPGL00004 is a potent allosteric glutaminase C (GAC) inhibitor (IC50=29 nM; Kd=27 nM)· UPGL00004 strongly inhibits the proliferation of highly aggressive triple-negative breast cancer cell lines
ChemicalCAS1890169-95-5MW534.66FormulaC25H26N8O2S2
- CAS number
- 1890169-95-5
- Molecular weight
- 534.66
- Formula
- C25H26N8O2S2
- Solubility
- DMSO： 125 mg/mL (233·79 mM)
- InChIKey
- MRYCNTHLPRENBA-UHFFFAOYSA-N
- Catalogue number
- GC61365
- Brand
- GLPBIO
Computed properties PubChem CID 121256411 · XLogP 4 · TPSA 182 Ų · H-bond donors 3
- XLogP
- 4
- TPSA
- 182 Ų
- H-bond donors
- 3
- H-bond acceptors
- 10
- Rotatable bonds
- 9
- Heavy atoms
- 37
SMILES C1CN(CCC1NC2=NN=C(S2)NC(=O)CC3=CC=CC=C3)C4=NN=C(S4)NC(=O)CC5=CC=CC=C5
Computed descriptors from PubChem (CID 121256411), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il