GC38653
Selumetinib sulfate
Also known as 6-(4-bromo-2-chloroanilino)-7-fluoro-N-(2-hydroxyethoxy)-3-methylbenzimidazole-5-carboxamide;sulfuric acid
Selumetinib (AZD6244) is selective, non-ATP-competitive oral?MEK1/2?inhibitor, with an IC50 of 14 nM for MEK1· Selumetinib (AZD6244) inhibits ERK1/2 phosphorylation
ChemicalCAS943332-08-9MW555.76FormulaC17H17BrClFN4O7S
- CAS number
- 943332-08-9
- Molecular weight
- 555.76
- Formula
- C17H17BrClFN4O7S
- Solubility
- DMSO： 50 mg/mL (89·97 mM); Water： ＜ 0·1 mg/mL (insoluble)
- InChIKey
- GRKFGZYYYYISDX-UHFFFAOYSA-N
- Catalogue number
- GC38653
- Brand
- GLPBIO
Computed properties PubChem CID 16214875 · TPSA 171 Ų · H-bond donors 5 · H-bond acceptors 10
- TPSA
- 171 Ų
- H-bond donors
- 5
- H-bond acceptors
- 10
- Rotatable bonds
- 6
- Heavy atoms
- 32
SMILES CN1C=NC2=C1C=C(C(=C2F)NC3=C(C=C(C=C3)Br)Cl)C(=O)NOCCO.OS(=O)(=O)O
Computed descriptors from PubChem (CID 16214875), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il