GC38501
GSK205
Also known as N-[4-[2-[benzyl(methyl)amino]ethyl]phenyl]-5-pyridin-3-yl-1,3-thiazol-2-amine;hydrobromide
GSK205 is a potent, selective TRPV4 antagonist with an IC50 of 4·19? μM for inhibiting TRPV4-mediated Ca2+ influx
ChemicalCAS1263068-83-2MW481.45FormulaC24H25BrN4S
- CAS number
- 1263068-83-2
- Molecular weight
- 481.45
- Formula
- C24H25BrN4S
- Solubility
- DMSO： 250 mg/mL (519·26 mM)
- InChIKey
- LQGOJHGNGSOUKL-UHFFFAOYSA-N
- Catalogue number
- GC38501
- Brand
- GLPBIO
Computed properties PubChem CID 72736243 · TPSA 69.3 Ų · H-bond donors 2 · H-bond acceptors 5
- TPSA
- 69.3 Ų
- H-bond donors
- 2
- H-bond acceptors
- 5
- Rotatable bonds
- 8
- Heavy atoms
- 30
SMILES CN(CCC1=CC=C(C=C1)NC2=NC=C(S2)C3=CN=CC=C3)CC4=CC=CC=C4.Br
Computed descriptors from PubChem (CID 72736243), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il