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Chemical structure of MT-802

GC36661

MT-802

Also known as 2-[2-[2-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]ethoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]acetamide

MT-802 is a potent BTK degrader based on Cereblon ligand, with a DC50 of 1 nM

ChemicalCAS2231744-29-7MW787.82FormulaC41H41N9O8
CAS number
2231744-29-7
Molecular weight
787.82
Formula
C41H41N9O8
Solubility
DMSO： 100 mg/mL (126·93 mM)
InChIKey
AJTLGUJXIKEZCQ-UHFFFAOYSA-N
Catalogue number
GC36661
Brand
GLPBIO
Computed properties PubChem CID 138108326 · XLogP 2.3 · TPSA 213 Ų · H-bond donors 3
XLogP
2.3
TPSA
213 Ų
H-bond donors
3
H-bond acceptors
13
Rotatable bonds
14
Heavy atoms
58

SMILES C1CC(=O)NC(=O)C1N2C(=O)C3=C(C2=O)C=C(C=C3)NC(=O)COCCOCCN4CCC(CC4)N5C6=NC=NC(=C6C(=N5)C7=CC=C(C=C7)OC8=CC=CC=C8)N

Computed descriptors from PubChem (CID 138108326), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
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Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.