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Chemical structure of Degarelix

GC35828

Degarelix

Also known as (4S)-N-[4-[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2R)-2-[[(2R)-2-acetamido-3-naphthalen-2-ylpropanoyl]amino]-3-(4-chlorophenyl)propanoyl]amino]-3-pyridin-3-ylpropanoyl]amino]-3-hydroxypropanoyl]amino]-3-[[(2R)-1-[[(2S)-1-[[(2S)-1-[(2S)-2-[[(2R)-1-amino-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxo-6-(propan-2-ylamino)hexan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-[4-(carbamoylamino)phenyl]-1-oxopropan-2-yl]amino]-3-oxopropyl]phenyl]-2,6-dioxo-1,3-diazinane-4-carboxamide

Degarelix is a competitive and reversible gonadotropin-releasing hormone receptor (GnRHR/LHRHR) antagonist

ChemicalCAS214766-78-6MW1632.26FormulaC82H103ClN18O16
CAS number
214766-78-6
Molecular weight
1632.26
Formula
C82H103ClN18O16
Solubility
Water： 25 mg/mL (15·32 mM); DMSO： 10 mg/mL (6·13 mM)
InChIKey
MEUCPCLKGZSHTA-XYAYPHGZSA-N
Catalogue number
GC35828
Brand
GLPBIO
Computed properties PubChem CID 16136245 · XLogP 3.5 · TPSA 513 Ų · H-bond donors 17
XLogP
3.5
TPSA
513 Ų
H-bond donors
17
H-bond acceptors
18
Rotatable bonds
41
Heavy atoms
117

SMILES C[C@H](C(=O)N)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCCNC(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC2=CC=C(C=C2)NC(=O)N)NC(=O)[C@H](CC3=CC=C(C=C3)NC(=O)[C@@H]4CC(=O)NC(=O)N4)NC(=O)[C@H](CO)NC(=O)[C@@H](CC5=CN=CC=C5)NC(=O)[C@@H](CC6=CC=C(C=C6)Cl)NC(=O)[C@@H](CC7=CC8=CC=CC=C8C=C7)NC(=O)C

Computed descriptors from PubChem (CID 16136245), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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