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Chemical structure of Conteltinib

GC35728

Conteltinib

Also known as 2-[[2-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]anilino]-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl]amino]-N-propan-2-ylbenzenesulfonamide

Conteltinib (CT-707) is a multi-kinase inhibitor targeting FAK, ALK, and Pyk2· Conteltinib exerts significant inhibitory effect on FAK with an IC50 of 1·6 nM

ChemicalCAS1384860-29-0MW635.82FormulaC32H45N9O3S
CAS number
1384860-29-0
Molecular weight
635.82
Formula
C32H45N9O3S
Solubility
DMSO： 31·25 mg/mL (49·15 mM)
InChIKey
NPJCURIANJMFEO-UHFFFAOYSA-N
Catalogue number
GC35728
Brand
GLPBIO
Computed properties PubChem CID 89860551 · XLogP 5.1 · TPSA 135 Ų · H-bond donors 4
XLogP
5.1
TPSA
135 Ų
H-bond donors
4
H-bond acceptors
12
Rotatable bonds
10
Heavy atoms
45

SMILES CC(C)NS(=O)(=O)C1=CC=CC=C1NC2=NC(=NC3=C2CCN3)NC4=C(C=C(C=C4)N5CCC(CC5)N6CCN(CC6)C)OC

Computed descriptors from PubChem (CID 89860551), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.