Loading...
Chemical structure of PROTAC BET-binding moiety 1

GC34725

PROTAC BET-binding moiety 1

Also known as 4-[(3-cyclopropyl-1-ethylpyrazol-5-yl)amino]-7-(3,5-dimethyl-1,2-oxazol-4-yl)-6-methoxy-9H-pyrimido[4,5-b]indole-2-carboxylic acid

PROTAC BET-binding moiety 1 is a key intermediate for the synthesis of high-affinity BET inhibitors

ChemicalCAS2093387-77-8MW487.51FormulaC25H25N7O4
CAS number
2093387-77-8
Molecular weight
487.51
Formula
C25H25N7O4
Solubility
Soluble in DMSO
InChIKey
DSICVZUZCUHARI-UHFFFAOYSA-N
Catalogue number
GC34725
Brand
GLPBIO
Computed properties PubChem CID 131988582 · XLogP 4.1 · TPSA 144 Ų · H-bond donors 3
XLogP
4.1
TPSA
144 Ų
H-bond donors
3
H-bond acceptors
9
Rotatable bonds
7
Heavy atoms
36

SMILES CCN1C(=CC(=N1)C2CC2)NC3=NC(=NC4=C3C5=CC(=C(C=C5N4)C6=C(ON=C6C)C)OC)C(=O)O

Computed descriptors from PubChem (CID 131988582), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.