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Chemical structure of RPR-260243

GC32509

RPR-260243

Also known as (3R,4R)-4-[3-(6-methoxyquinolin-4-yl)-3-oxopropyl]-1-[3-(2,3,5-trifluorophenyl)prop-2-ynyl]piperidine-3-carboxylic acid

RPR-260243, a potent activator of human ether-a-go-go-related gene (hERG), slows deactivation and attenuates inactivation of hERG1 channels

ChemicalCAS668463-35-2MW510.5FormulaC28H25F3N2O4
CAS number
668463-35-2
Molecular weight
510.5
Formula
C28H25F3N2O4
Solubility
DMSO： 10 mg/mL (19·59 mM)
InChIKey
VWNMWKSURFWKAL-HXOBKFHXSA-N
Catalogue number
GC32509
Brand
GLPBIO
Computed properties PubChem CID 11466357 · XLogP 2 · TPSA 79.7 Ų · H-bond donors 1
XLogP
2
TPSA
79.7 Ų
H-bond donors
1
H-bond acceptors
9
Rotatable bonds
8
Heavy atoms
37

SMILES COC1=CC2=C(C=CN=C2C=C1)C(=O)CC[C@@H]3CCN(C[C@@H]3C(=O)O)CC#CC4=C(C(=CC(=C4)F)F)F

Computed descriptors from PubChem (CID 11466357), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

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