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Chemical structure of RG3039 (PF-06687859)

GC30784

RG3039 (PF-06687859)

Also known as 5-[[1-[(2,6-dichlorophenyl)methyl]piperidin-4-yl]methoxy]quinazoline-2,4-diamine

RG3039 (PF-06687859) (PF-06687859) is an orally bioavailable and brain-penetrant DcpS inhibitor with an IC50 of 0·069 nM

ChemicalCAS1005504-62-0MW432.35FormulaC21H23Cl2N5O
CAS number
1005504-62-0
Molecular weight
432.35
Formula
C21H23Cl2N5O
Solubility
DMSO ： 6 mg/mL (13·88 mM);Water ： ＜ 0·1 mg/mL (insoluble)
InChIKey
MNLHFGXIUJNDAF-UHFFFAOYSA-N
Catalogue number
GC30784
Brand
GLPBIO
Computed properties PubChem CID 53258905 · XLogP 4.3 · TPSA 90.3 Ų · H-bond donors 2
XLogP
4.3
TPSA
90.3 Ų
H-bond donors
2
H-bond acceptors
6
Rotatable bonds
5
Heavy atoms
29

SMILES C1CN(CCC1COC2=CC=CC3=C2C(=NC(=N3)N)N)CC4=C(C=CC=C4Cl)Cl

Computed descriptors from PubChem (CID 53258905), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.