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Chemical structure of EEDi-5273

GC26751

EEDi-5273

Also known as 15-[(5-fluoro-2,3-dihydro-1-benzofuran-4-yl)methylamino]-9-propan-2-yl-5-(trifluoromethyl)-4,9,12,14,16-pentazatetracyclo[9.6.1.02,7.014,18]octadeca-1(17),2,4,6,11(18),12,15-heptaen-10-one

EEDi-5273 is an exceptionally potent and orally efficacious EED inhibitor (IC50 = 0·2 nM) capable of achieving complete and persistent tumor regression

ChemicalCAS2585648-55-9MW526.49FormulaC26H22F4N6O2
CAS number
2585648-55-9
Molecular weight
526.49
Formula
C26H22F4N6O2
Solubility
DMSO ： 25 mg/mL (47·48 mM; Need ultrasonic)
InChIKey
OAYMRNSLBKYMKG-UHFFFAOYSA-N
Catalogue number
GC26751
Brand
GLPBIO
Computed properties PubChem CID 155580034 · XLogP 4.8 · TPSA 84.7 Ų · H-bond donors 1
XLogP
4.8
TPSA
84.7 Ų
H-bond donors
1
H-bond acceptors
10
Rotatable bonds
4
Heavy atoms
38

SMILES CC(C)N1CC2=CC(=NC=C2C3=CN=C(N4C3=C(C1=O)N=C4)NCC5=C(C=CC6=C5CCO6)F)C(F)(F)F

Computed descriptors from PubChem (CID 155580034), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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