Loading...
Chemical structure of Varenicline (CP 526555) dihydrochloride

GC26032

Varenicline (CP 526555) dihydrochloride

Also known as 5,8,14-triazatetracyclo[10.3.1.02,11.04,9]hexadeca-2,4,6,8,10-pentaene;dihydrochloride

Varenicline (CP 526555, Chantix, Champix,CP 526555 dihydrochloride) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR with EC50 of 2·3 μM and 55 μM, respectively· Varenicline dihydrochloride is a potent, full agonist of α7 nAChRs with EC50 of 18 μM· Varenicline is a prescription medication used for smoking cessation

ChemicalCAS866823-63-4MW284.18FormulaC13H15Cl2N3
CAS number
866823-63-4
Molecular weight
284.18
Formula
C13H15Cl2N3
Solubility
DMSO： 57 mg/mL (200·58 mM);Water： 57 mg/mL (200·58 mM);Ethanol： 29 mg/mL (102·05 mM)
InChIKey
NZVVYNGXLGJKCW-UHFFFAOYSA-N
Catalogue number
GC26032
Brand
GLPBIO
Computed properties PubChem CID 45263226 · TPSA 37.8 Ų · H-bond donors 3 · H-bond acceptors 3
TPSA
37.8 Ų
H-bond donors
3
H-bond acceptors
3
Rotatable bonds
0
Heavy atoms
18

SMILES C1C2CNCC1C3=CC4=NC=CN=C4C=C23.Cl.Cl

Computed descriptors from PubChem (CID 45263226), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.