GC25982
Tanzisertib(CC-930)
Tanzisertib (CC-930, JNK-930, JNKI-1) is kinetically competitive with ATP in the JNK-dependent phosphorylation of the protein substrate c-Jun and potent against all isoforms of JNK (Ki(JNK1) = 44 ± 3 nM, IC50(JNK1) = 61 nM, Ki(JNK2) = 6·2 ± 0·6 nM, IC50(JNK2) = 5 nM, IC50(JNK3) = 5 nM) and selective against MAP kinases ERK1 and p38a with IC50 of 0·48 and 3·4 μM respectively
ChemicalMW484.9FormulaC21H23F3N6O2·HCl
- CAS number
- —
- Molecular weight
- 484.9
- Formula
- C21H23F3N6O2·HCl
- Solubility
- DMSO： 89 mg/mL (183·54 mM);Water： 4 mg/mL (8·25 mM);Ethanol： 89 mg/mL (183·54 mM)
- Catalogue number
- GC25982
- Brand
- GLPBIO
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il