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Chemical structure of LP99

GC18731

LP99

Also known as N-[(2R,3S)-2-(4-chlorophenyl)-1-(1,4-dimethyl-2-oxoquinolin-7-yl)-6-oxopiperidin-3-yl]-2-methylpropane-1-sulfonamide

LP99 is a potent inhibitor of the bromodomain containing proteins BRD7 and BRD9 that binds with Kd values of 99 and 909 nM, respectively, as determined by isothermal titration calorimetry

ChemicalCAS1808951-93-0MW516.1FormulaC26H30ClN3O4S
CAS number
1808951-93-0
Molecular weight
516.1
Formula
C26H30ClN3O4S
Solubility
DMF： 20 mg/ml,DMSO： 20 mg/ml,Ethanol： 20 mg/ml,Ethanol：PBS (pH 7·2) (1：9)： 0·1 mg/ml
InChIKey
LVDRREOUMKACNJ-BKMJKUGQSA-N
Catalogue number
GC18731
Brand
GLPBIO
Computed properties PubChem CID 91827372 · XLogP 3.5 · TPSA 95.2 Ų · H-bond donors 1
XLogP
3.5
TPSA
95.2 Ų
H-bond donors
1
H-bond acceptors
5
Rotatable bonds
6
Heavy atoms
35

SMILES CC1=CC(=O)N(C2=C1C=CC(=C2)N3[C@@H]([C@H](CCC3=O)NS(=O)(=O)CC(C)C)C4=CC=C(C=C4)Cl)C

Computed descriptors from PubChem (CID 91827372), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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