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Chemical structure of SCH772984

GC16001

SCH772984

Also known as (3R)-1-[2-oxo-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-N-(3-pyridin-4-yl-1H-indazol-5-yl)pyrrolidine-3-carboxamide

SCH772984 is a novel, potent, ATP-competitive inhibitor of ERK1 and ERK2 with IC50 values of 4nM and 1nM, respectively

ChemicalCAS942183-80-4MW587.67FormulaC33H33N9O2
CAS number
942183-80-4
Molecular weight
587.67
Formula
C33H33N9O2
Solubility
≥ 14·7 mg/mL in DMSO with gentle warming
InChIKey
HDAJDNHIBCDLQF-RUZDIDTESA-N
Catalogue number
GC16001
Brand
GLPBIO
Computed properties PubChem CID 24866313 · XLogP 2.5 · TPSA 123 Ų · H-bond donors 2
XLogP
2.5
TPSA
123 Ų
H-bond donors
2
H-bond acceptors
8
Rotatable bonds
7
Heavy atoms
44

SMILES C1CN(C[C@@H]1C(=O)NC2=CC3=C(C=C2)NN=C3C4=CC=NC=C4)CC(=O)N5CCN(CC5)C6=CC=C(C=C6)C7=NC=CC=N7

Computed descriptors from PubChem (CID 24866313), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.