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Chemical structure of AM251

GC15717

AM251

Also known as 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide

AM251 is a cannabinoid receptor type 1 (CB1) antagonist with an IC50 of 8nM and a G protein-coupled receptor 55 (GPR55) agonist with an EC50 of 39nM

ChemicalCAS183232-66-8MW555.24FormulaC22H21Cl2IN4O
CAS number
183232-66-8
Molecular weight
555.24
Formula
C22H21Cl2IN4O
Solubility
≥ 55·5mg/mL in DMSO with gentle warming
InChIKey
BUZAJRPLUGXRAB-UHFFFAOYSA-N
Catalogue number
GC15717
Brand
GLPBIO
Computed properties PubChem CID 2125 · XLogP 6.5 · TPSA 50.2 Ų · H-bond donors 1
XLogP
6.5
TPSA
50.2 Ų
H-bond donors
1
H-bond acceptors
3
Rotatable bonds
4
Heavy atoms
30

SMILES CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)I

Computed descriptors from PubChem (CID 2125), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
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Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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