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Chemical structure of GI 254023X

GC14578

GI 254023X

Also known as (2R)-N-[(2S)-3,3-dimethyl-1-(methylamino)-1-oxobutan-2-yl]-2-[(1S)-1-[formyl(hydroxy)amino]ethyl]-5-phenylpentanamide

GI 254023X is a selective inhibitor with an IC50 value of 5·3nM for MMP9 (Matrix Metalloproteinase 9)· The selectivity of GI 254023X for ADAM10 (A Disintegrin and Metalloproteinase 10) is 100 times higher than that for ADAM17, with an IC50 value of 2·5nM· GI 254023X is primarily used in the research of immunology, inflammation, and neurodegenerative diseases

ChemicalCAS260264-93-5MW391.5FormulaC21H33N3O4
CAS number
260264-93-5
Molecular weight
391.5
Formula
C21H33N3O4
Solubility
DMF： 1 mg/mL,Ethanol： 1 mg/mL,Ethanol：PBS (pH 7·2) (1：6)： 0·14mg/mL
InChIKey
GHVMTHKJUAOZJP-CGTJXYLNSA-N
Catalogue number
GC14578
Brand
GLPBIO
Computed properties PubChem CID 9952396 · XLogP 2.9 · TPSA 98.7 Ų · H-bond donors 3
XLogP
2.9
TPSA
98.7 Ų
H-bond donors
3
H-bond acceptors
4
Rotatable bonds
10
Heavy atoms
28

SMILES C[C@@H]([C@@H](CCCC1=CC=CC=C1)C(=O)N[C@H](C(=O)NC)C(C)(C)C)N(C=O)O

Computed descriptors from PubChem (CID 9952396), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.