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Chemical structure of RVX-208

GC14199

RVX-208

Also known as 2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-5,7-dimethoxy-3H-quinazolin-4-one

RVX-208 (RVX-208) is an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain· The IC50s are 87 μM and 0·51 μM for BD1 and BD2, respectively

ChemicalCAS1044870-39-4MW370.4FormulaC20H22N2O5
CAS number
1044870-39-4
Molecular weight
370.4
Formula
C20H22N2O5
Solubility
≥ 18·52mg/mL in DMSO
InChIKey
NETXMUIMUZJUTB-UHFFFAOYSA-N
Catalogue number
GC14199
Brand
GLPBIO
Computed properties PubChem CID 135564749 · XLogP 2.3 · TPSA 89.4 Ų · H-bond donors 2
XLogP
2.3
TPSA
89.4 Ų
H-bond donors
2
H-bond acceptors
6
Rotatable bonds
6
Heavy atoms
27

SMILES CC1=CC(=CC(=C1OCCO)C)C2=NC3=C(C(=CC(=C3)OC)OC)C(=O)N2

Computed descriptors from PubChem (CID 135564749), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

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