GC12952
PNU 282987
PNU 282987 is a selective α7 nicotinic acetylcholine receptor (α7nAChR) agonist associated with an anti-inflammatory pathway as well as an antagonist of the 5-HT3 receptor, the EC50 of PNU 282987 for α7nAChR is 154nM (Ki α7nAChR=27nM, rat brain homogenates) while IC50 for 5-HT3 receptor is 4541nM (Ki 5-HT3R=1662nM, GR-65630)
ChemicalCAS123464-89-1MW264.75FormulaC14H17ClN2O
- CAS number
- 123464-89-1
- Molecular weight
- 264.75
- Formula
- C14H17ClN2O
- Solubility
- DMF： 10 mg/ml,DMSO： 30 mg/ml,Ethanol： 20 mg/ml,PBS (pH 7·2)： 5 mg/ml
- Catalogue number
- GC12952
- Brand
- GLPBIO
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il