
GC12667
4SC-202
Also known as (E)-N-(2-aminophenyl)-3-[1-[4-(1-methylpyrazol-4-yl)phenyl]sulfonylpyrrol-3-yl]prop-2-enamide;4-methylbenzenesulfonic acid
4SC-202 (4SC-202) is a selective class I HDAC inhibitor with IC50 of 1·20 μM, 1·12 μM, and 0·57 μM for HDAC1, HDAC2, and HDAC3, respectively· It also displays inhibitory activity against Lysine specific demethylase 1 (LSD1)
ChemicalCAS1186222-89-8MW619.71FormulaC30H29N5O6S2
- CAS number
- 1186222-89-8
- Molecular weight
- 619.71
- Formula
- C30H29N5O6S2
- Solubility
- ≥ 62mg/mL in DMSO
- InChIKey
- IAVXAZDVNICKFJ-ICSBZGNSSA-N
- Catalogue number
- GC12667
- Brand
- GLPBIO
Computed properties PubChem CID 44217246 · TPSA 183 Ų · H-bond donors 3 · H-bond acceptors 8
- TPSA
- 183 Ų
- H-bond donors
- 3
- H-bond acceptors
- 8
- Rotatable bonds
- 7
- Heavy atoms
- 43
SMILES CC1=CC=C(C=C1)S(=O)(=O)O.CN1C=C(C=N1)C2=CC=C(C=C2)S(=O)(=O)N3C=CC(=C3)/C=C/C(=O)NC4=CC=CC=C4N
Computed descriptors from PubChem (CID 44217246), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il