
GB40167
D 106669
Also known as 1-ethyl-3-[3-(4-methylanilino)pyrido[2,3-b]pyrazin-6-yl]urea
Highly potent and selective PI3K inhibitor, selectively inhibiting class I PI3K (PI3Kα IC50 3 log selectivity against tyrosine or serine/threonine kinases, except ERK1 and 2) and showed some activity in A549 (lung cancer) xenografts mouse model at oral dose of 30 mg/kg twice daily
ChemicalCAS938444-93-0MW322.36FormulaC17H18N6O
- CAS number
- 938444-93-0
- Molecular weight
- 322.36
- Formula
- C17H18N6O
- InChIKey
- RQBRFKKFZPOBFG-UHFFFAOYSA-N
- Catalogue number
- GB40167
- Brand
- GLPBIO
Computed properties PubChem CID 16048654 · XLogP 2.4 · TPSA 91.8 Ų · H-bond donors 3
- XLogP
- 2.4
- TPSA
- 91.8 Ų
- H-bond donors
- 3
- H-bond acceptors
- 5
- Rotatable bonds
- 4
- Heavy atoms
- 24
SMILES CCNC(=O)NC1=NC2=NC(=CN=C2C=C1)NC3=CC=C(C=C3)C
Computed descriptors from PubChem (CID 16048654), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il