GB40105
AT 1001
High affinity and selective α3β4 nAChR ligand (Ki value 2·6 nM at α3β4 nAChR) with both partial agonistic and antagonistic effects, and >90-fold selective over the other major subtypes, the α4β2 and α7 nAChR· AT-1001 potently and dose-dependently blocks nicotine self-administration in rats, without affecting food responding, and shows a mechanism of action very different from varenicline (Varenicline dihydrochloride (HCl salt) and AT 1001 (tartrate salt))
ChemicalCAS1314801-63-2MW309.24FormulaC15H21BrN2
- CAS number
- 1314801-63-2
- Molecular weight
- 309.24
- Formula
- C15H21BrN2
- Catalogue number
- GB40105
- Brand
- GLPBIO
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il