
GA22966
H-Tyr-Cys-Phe-Ala-Trp-Lys-Thr-Phe-Cys-OH
Selective somatostatin receptor subtype sst4 agonist· In competitive radioligand displacement experiments using the non-selective radioligand ([¹²?I]-(Leu?,D-Trp²²,Tyr²?)-Somatostatin-28, YCFAWKTFC exhibited a high affinity for sst4 with an IC?? value of 2·0 ± 0·5 nM· IC?? values for sst1, sst2, sst3, and sst5 were >1000 nM, 622 ± 85 nM, 624 ± 213 nM, and 692 ± 166 nM, respectively· The nonapeptide YCFAWKTFC may serve as a lead compound or tool for preclinical and clinical studies
ChemicalCAS647016-22-6MW1166.39FormulaC57H71N11O12S2
- CAS number
- 647016-22-6
- Molecular weight
- 1166.39
- Formula
- C57H71N11O12S2
- Solubility
- Soluble in DMSO
- Catalogue number
- GA22966
- Brand
- GLPBIO
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il