
GA22468
H-Gly-His-Arg-Pro-NH₂
Also known as (2S)-1-[(2S)-2-[[(2S)-2-[(2-aminoacetyl)amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carboxamide
The central E region of fibrin contains two sets of polymerization knobs, A and B, that are cryptic in fibrinogen but become exposed after thrombin cleavage of fibrinopeptide A (FpA) and fibrinopeptide B (FpB) from the N-terminus of the Aα- and Bβ-chains, respectively· The location of the binding holes and possible models for knob-hole interactions are known from X-ray crystallographic studies using synthetic peptide analogs of knobs A and B· When fibrinogen fragment D and double-D are crystallized in the presence of both peptide analogs, the knob A peptide mimic H-Gly-Pro-Arg-Pro-NH? (GPRP-amide, H-1998) forms H-bond interactions with residues γ364Asp, γ330Asp, γ329Gln, and γ340His found in hole a· In the same manner, the knob B peptide mimic H-Gly-His-Arg-Pro-NH? (GHRP-amide, H-7318) interacts with residues Bβ397Glu, Bβ398Asp, and Bβ432Asp in hole b
- CAS number
- 209623-54-1
- Molecular weight
- 464.53
- Formula
- C19H32N10O4
- Solubility
- Soluble in DMSO
- InChIKey
- FFSSGCULYCDLRM-IHRRRGAJSA-N
- Catalogue number
- GA22468
- Brand
- GLPBIO
Computed properties PubChem CID 447016 · XLogP -4.3 · TPSA 241 Ų · H-bond donors 7
- XLogP
- -4.3
- TPSA
- 241 Ų
- H-bond donors
- 7
- H-bond acceptors
- 7
- Rotatable bonds
- 12
- Heavy atoms
- 33
SMILES C1C[C@H](N(C1)C(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CC2=CN=CN2)NC(=O)CN)C(=O)N
Computed descriptors from PubChem (CID 447016), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il