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Chemical structure of H-Glu[cyclo(-Arg-Gly-Asp-D-Phe-Lys)]-cyclo(-Arg-Gly-Asp-D-Phe-Lys)

GA22370

H-Glu[cyclo(-Arg-Gly-Asp-D-Phe-Lys)]-cyclo(-Arg-Gly-Asp-D-Phe-Lys)

Also known as 2-[(2S,5R,8S,11S)-8-[4-[[(4S)-4-amino-5-[4-[(2S,5S,11S,14R)-14-benzyl-11-(carboxymethyl)-5-[3-(diaminomethylideneamino)propyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]butylamino]-5-oxopentanoyl]amino]butyl]-5-benzyl-11-[3-(diaminomethylideneamino)propyl]-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]acetic acid

E(c(RGDfK))? (SU 016), a dimeric form of c(RGDfK), showed improved tumor targeting properties compared to the monomer· E(c(RGDfK))? can be easily conjugated to dyes, drug molecules, or chelators· The ??Ga complex of DOTA-E(c(RGDfK))? has been evaluated as theranostic radiopharmaceutical

ChemicalCAS250612-47-6MW1318.46FormulaC59H87N19O16
CAS number
250612-47-6
Molecular weight
1318.46
Formula
C59H87N19O16
Solubility
Soluble in DMSO
InChIKey
HBRYUNRKUGWZGH-LMKMLFLWSA-N
Catalogue number
GA22370
Brand
GLPBIO
Computed properties PubChem CID 59045268 · XLogP -7.3 · TPSA 579 Ų · H-bond donors 19
XLogP
-7.3
TPSA
579 Ų
H-bond donors
19
H-bond acceptors
19
Rotatable bonds
30
Heavy atoms
94

SMILES C1C(=O)N[C@H](C(=O)N[C@@H](C(=O)N[C@H](C(=O)N[C@H](C(=O)N1)CCCN=C(N)N)CCCCNC(=O)CC[C@@H](C(=O)NCCCC[C@H]2C(=O)N[C@H](C(=O)NCC(=O)N[C@H](C(=O)N[C@@H](C(=O)N2)CC3=CC=CC=C3)CC(=O)O)CCCN=C(N)N)N)CC4=CC=CC=C4)CC(=O)O

Computed descriptors from PubChem (CID 59045268), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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