
GA20281
(Propionyl¹,D-Tyr(Et)²,Val⁴,Abu⁶,Arg⁸,⁹)-Vasopressin
Also known as (2S)-N-[(2S)-1-[(2S)-2-[[(2S)-1-[[(2S)-1-amino-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1-oxobutan-2-yl]-2-[[(2S)-2-[[(2S)-2-[[(2R)-3-(4-ethoxyphenyl)-2-(propanoylamino)propanoyl]amino]-3-phenylpropanoyl]amino]-3-methylbutanoyl]amino]butanediamide
This linear vasopressin analog is as potent a V? (antidiuretic) antagonist as its cyclic parent compound· Its V? (vasopressor) antagonism, however, is significantly reduced, resulting in a promising anti-V?/anti-V? selectivity
- CAS number
- 121250-95-1
- Molecular weight
- 1119.34
- Formula
- C53H82N16O11
- Solubility
- Soluble in DMSO
- InChIKey
- MVBVPHFFZQUTBB-RIKPAVIRSA-N
- Catalogue number
- GA20281
- Brand
- GLPBIO
Computed properties PubChem CID 14310031 · XLogP -1 · TPSA 448 Ų · H-bond donors 13
- XLogP
- -1
- TPSA
- 448 Ų
- H-bond donors
- 13
- H-bond acceptors
- 13
- Rotatable bonds
- 34
- Heavy atoms
- 80
SMILES CC[C@@H](C(=O)N1CCC[C@H]1C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N)NC(=O)[C@H](CC(=O)N)NC(=O)[C@H](C(C)C)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@@H](CC3=CC=C(C=C3)OCC)NC(=O)CC
Computed descriptors from PubChem (CID 14310031), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il